Comprehensive Survey of Combinatorial Library Synthesis:  2001

The Design of Leadlike Combinatorial Libraries

Simon J. Teague, A. M. Davis, Paul D. Leeson et al. · Angewandte Chemie International Edition · 1999 · 810 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17

Is There a Difference between Leads and Drugs? A Historical Perspective

Tudor I. Oprea, A. M. Davis, Simon J. Teague et al. · Journal of Chemical Information and Computer Sciences · 2001 · 775 citations

Pharmacy, Medicinal Chemistry, Pharmacology +12

Automated Library Generation Using Sequential Microwave-Assisted Chemistry. Application toward the Biginelli Multicomponent Condensation

Alexander Stadler, C. Oliver Kappe · Journal of Combinatorial Chemistry · 2001 · 232 citations

Pharmacy, Chemical Engineering, Chemistry +14

Global analysis of proteasomal substrate specificity using positional-scanning libraries of covalent inhibitors

Tamim Nazif, Matthew Bogyo · Proceedings of the National Academy of Sciences · 2001 · 179 citations · Full text

Life Sciences, Biochemistry, Molecular Biology +17

Novel procedure for the synthesis of 1,3,4-oxadiazoles from 1,2-diacylhydrazines using polymer-supported Burgess reagent under microwave conditions

Christopher T. Brain, Jane M. Paul, Yvonne Loong et al. · Tetrahedron Letters · 1999 · 179 citations

Natural Sciences, Chemistry, Organic Chemistry +8