Concepedia

Design and synthesis of a biaryl series as inhibitors for the bromodomains of CBP/P300

Kwong Wah Lai, F. Anthony Romero, Vickie Tsui, Maureen H. Beresini, Gladys de Leon Boenig, Sarah M. Bronner, Kevin Chen, Zhongguo Chen, Edna F. Choo, Terry D. Crawford,

Bioorganic & Medicinal Chemistry Letters · 2017 · 31 citations · 27 references

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References

27

The Transcriptional Coactivators p300 and CBP Are Histone Acetyltransferases

Vasily Ogryzko, R. Louis Schiltz, Valya Russanova et al. · Cell · 1996 · 3K citations · Full text

, , +13

The CBP co-activator is a histone acetyltransferase

Andrew J. Bannister, Tony Kouzarides · Nature · 1996 · 1.8K citations

, , +11

Solution Structure of the KIX Domain of CBP Bound to the Transactivation Domain of CREB: A Model for Activator:Coactivator Interactions

Ishwar Radhakrishnan, Gabriela C. Pérez-Alvarado, David Parker et al. · Cell · 1997 · 730 citations · Full text

, , +13

p300/CBP‐mediated p53 acetylation is commonly induced by p53‐activating agents and inhibited by MDM2

Akihiro Ito, Chun-Hsiang Lai, Xuan Zhao et al. · The EMBO Journal · 2001 · 575 citations · Full text

, , +4

Aromatic–Proline Interactions: Electronically Tunable CH/π Interactions

Neal J. Zondlo · Accounts of Chemical Research · 2012 · 321 citations

, , +17