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A comparative study of warheads for design of cysteine protease inhibitors

Daniel Giura da Silva, Jean F. R. Ribeiro, Daniela De Vita, Lorenzo Cianni, Caio Haddad Franco, Lúcio H. Freitas-Júnior, Carolina Borsoi Moraes, Josmar R. Rocha, Antonio C. B. Burtoloso, Peter W. Kenny,

Bioorganic & Medicinal Chemistry Letters · 2017 · 53 citations · 19 references

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Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design

Nicholas A. Meanwell · Journal of Medicinal Chemistry · 2011 · 2.8K citations · Full text

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The discovery of odanacatib (MK-0822), a selective inhibitor of cathepsin K

Jacques Yves Gauthier, Nathalie Chauret, Wanda Cromlish et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 473 citations · Full text

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Nitroheterocyclic compounds are more efficacious than CYP51 inhibitors against Trypanosoma cruzi: implications for Chagas disease drug discovery and development

Carolina Borsoi Moraes, Miriam A. Giardini, Hwayoung Kim et al. · Scientific Reports · 2014 · 208 citations · Full text

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Cysteine protease inhibitors as chemotherapy: Lessons from a parasite target

Paul M. Selzer, Sabine Pingel, Ivy Hsieh et al. · Proceedings of the National Academy of Sciences · 1999 · 193 citations · Full text

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Hydrogen Bonding, Electrostatic Potential, and Molecular Design

Peter W. Kenny · Journal of Chemical Information and Modeling · 2009 · 167 citations

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