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Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings

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From the Triumvirate to the Ominous Octet: A New Paradigm for the Treatment of Type 2 Diabetes Mellitus

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Immunology, Insulin Signaling, Metabolic Syndrome +17

Microvascular and Macrovascular Complications of Diabetes

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Type 1, Diabetic Retinopathy, Diabetes Management +14

Free fatty acids regulate insulin secretion from pancreatic β cells through GPR40

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Metabolic Syndrome, Insulin Signaling, Molecular Physiology +14

Principles and Applications of Halogen Bonding in Medicinal Chemistry and Chemical Biology

Rainer Wilcken, Markus O. Zimmermann, Andreas Lange et al. · Journal of Medicinal Chemistry · 2012 · 1.3K citations · Full text

Halogenation, Molecular Recognition, Medicinal Chemistry +15