Target Residence Time-Guided Optimization on TTK Kinase Results in Inhibitors with Potent Anti-Proliferative Activity

Joost C.M. Uitdehaag, Jos de Man, Nicole Willemsen‐Seegers, Martine B.W. Prinsen, Marion A.A. Libouban, Jan Gerard Sterrenburg, Joeri J.P. de Wit, Judith R.F. de Vetter, Jeroen A.D.M. de Roos, Rogier C. Buijsman,

Journal of Molecular Biology · 2017 · 63 citations · 42 references

Concepts

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