Kinetic resolution of vinyl carbonates through a lipase-mediated synthesis of their carbonate and carbamate derivatives.

N,N`-dissuccinimidyl carbonate: a useful reagent for alkoxycarbonylation of amines

Arun K. Ghosh, Tien T. Doung, S. P. MCKEE et al. · Tetrahedron Letters · 1992 · 97 citations · Full text

Natural Sciences, Chemistry, Medicinal Chemistry +4

Selective delivery of cytotoxic compounds to cells by the LDL pathway

Raymond A. Firestone, Judith M. Pisano, John R. Falck et al. · Journal of Medicinal Chemistry · 1984 · 93 citations

Life Sciences, Biochemistry, Pharmacology +17

Evolution of a series of peptidoleukotriene antagonists: synthesis and structure-activity relationships of 1,6-disubstituted indoles and indazoles

F.J. Brown, Ying K. Yee, Laura A. Cronk et al. · Journal of Medicinal Chemistry · 1990 · 89 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +12

(Acyloxy)alkyl carbamates as novel bioreversible prodrugs for amines: increased permeation through biological membranes

Jose Alexander, Robyn Cargill, Stuart R. Michelson et al. · Journal of Medicinal Chemistry · 1988 · 83 citations

Pharmacy, Medicinal Chemistry, Pharmacology +11

Evolution of a series of peptidoleukotriene antagonists: synthesis and structure/activity relationships of 1,3,5-substituted indoles and indazoles

Victor G. Matassa, Thomas Maduskuie, Howard S. Shapiro et al. · Journal of Medicinal Chemistry · 1990 · 78 citations

Pharmacy, Medicinal Chemistry, Pharmacology +12