Stuart R. Michelson

Design and Synthesis of 8-Hydroxy-[1,6]Naphthyridines as Novel Inhibitors of HIV-1 Integrase in Vitro and in Infected Cells

Linghang Zhuang, John Wai, Mark W. Embrey et al. · Journal of Medicinal Chemistry · 2003 · 270 citations · Full text

Pharmacy, Pharmacokinetics, Pharmacology +17

New isomeric classes of topically active ocular hypotensive carbonic anhydrase inhibitors: 5-substituted thieno[2,3-b]thiophene-2-sulfonamides and 5-substituted thieno[3,2-b]thiophene-2-sulfonamides

John D. Prugh, George D. Hartman, Pierre Mallorga et al. · Journal of Medicinal Chemistry · 1991 · 117 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +10

(Acyloxy)alkyl carbamates as novel bioreversible prodrugs for amines: increased permeation through biological membranes

Jose Alexander, Robyn Cargill, Stuart R. Michelson et al. · Journal of Medicinal Chemistry · 1988 · 83 citations

Pharmacy, Medicinal Chemistry, Pharmacology +11

Development of Orally Active Oxytocin Antagonists:  Studies on 1-(1-{4-[1-(2-Methyl-1-oxidopyridin-3-ylmethyl)piperidin-4-yloxy]-2- methoxybenzoyl}piperidin-4-yl)-1,4-dihydrobenz[<i>d</i>][1,3]oxazin-2-one (L-372,662) and Related Pyridines

Ian M. Bell, Jill M. Erb, Roger Freidinger et al. · Journal of Medicinal Chemistry · 1998 · 60 citations · Full text

Pharmacy, Pharmacokinetics, Pharmacology +13

Affinity purification of the HIV-1 protease

Jill C. Heimbach, Victor M. Garsky, Stuart R. Michelson et al. · Biochemical and Biophysical Research Communications · 1989 · 58 citations

Life Sciences, Biochemistry, Molecular Biology +14