In vivo pharmacology of ICI 198,615: a novel, potent and selective peptide leukotriene antagonist.

Robert D. Krell, Ralph E. Giles, Ying K. Yee, +1

Journal of Pharmacology and Experimental Therapeutics

Identification of Essential Residues for the Catalytic Function of 85-kDa Cytosolic Phospholipase A2

Richard T. Pickard, X. Grace Chiou, Beth A. Strifler, +8

Journal of Biological Chemistry

Evolution of a series of peptidoleukotriene antagonists: synthesis and structure-activity relationships of 1,6-disubstituted indoles and indazoles

F.J. Brown, Ying K. Yee, Laura A. Cronk, +3

Journal of Medicinal Chemistry

A novel series of selective leukotriene antagonists: exploration and optimization of the acidic region in 1,6-disubstituted indoles and indazoles

Ying K. Yee, Peter R Bernstein, Edward J. Adams, +6

Journal of Medicinal Chemistry

Pharmaceutical ScienceSystematic Structure-activity ExplorationPharmacotherapyHeterocycle ChemistryAcid 1 +15

Conjugate and direct addition of ester enolates to cyclohexenone. Selective control of reaction composition

Arthur G. Schultz, Ying K. Yee

The Journal of Organic Chemistry

Reaction CompositionEngineeringEnantioselective SynthesisBiochemistryNatural Sciences +10

Novel 3-Aryl Indoles as Progesterone Receptor Antagonists for Uterine Fibroids

Timothy I. Richardson, Christian A. Clarke, Kuo‐Long Yu, +16

ACS Medicinal Chemistry Letters

Medicinal ChemistryHormonal ContraceptiveUterine FibroidsProgesterone AntagonismBiochemistry +13

<i>N</i>²-Aroylanthranilamide Inhibitors of Human Factor Xa

Ying K. Yee, Anne Louise Tebbe, Jared H. Linebarger, +13

Journal of Medicinal Chemistry

Molecular PharmacologyMedicinal ChemistryDrug TargetHfxa KBiochemistry +12

Structure-Based Design of Potent, Amidine-Derived Inhibitors of Factor Xa:  Evaluation of Selectivity, Anticoagulant Activity, and Antithrombotic Activity

Michael R. Wiley, Leonard C. Weir, Steven L. Briggs, +26

Journal of Medicinal Chemistry

Drug TargetPharmacotherapyAmidine-derived InhibitorsChemical BiologyPharmaceutical Chemistry +18

Hydroxyacetophenone-derived antagonists of the peptidoleukotrienes

Frederick J. Brown, Peter R Bernstein, Laura A. Cronk, +6

Journal of Medicinal Chemistry

Medicinal ChemistryPharmaceutical ScienceBiochemistryMedicineNatural Sciences +11

Non-Amidine-Containing 1,2-Dibenzamidobenzene Inhibitors of Human Factor Xa with Potent Anticoagulant and Antithrombotic Activity

John J. Masters, Jeffry B. Franciskovich, Jennifer M. Tinsley, +18

Journal of Medicinal Chemistry

Altmetric Attention ScorePharmacotherapyTranslational PharmacologyPre-clinical PharmacologyThrombosis +17