Laura A. Cronk

Evolution of a series of peptidoleukotriene antagonists: synthesis and structure-activity relationships of 1,6-disubstituted indoles and indazoles

F.J. Brown, Ying K. Yee, Laura A. Cronk et al. · Journal of Medicinal Chemistry · 1990 · 89 citations · Full text

A novel series of selective leukotriene antagonists: exploration and optimization of the acidic region in 1,6-disubstituted indoles and indazoles

Ying K. Yee, Peter R Bernstein, Edward J. Adams et al. · Journal of Medicinal Chemistry · 1990 · 60 citations

Pharmaceutical Science, Systematic Structure-activity Exploration, Pharmacotherapy +17

Hydroxyacetophenone-derived antagonists of the peptidoleukotrienes

Frederick J. Brown, Peter R Bernstein, Laura A. Cronk et al. · Journal of Medicinal Chemistry · 1989 · 44 citations

Medicinal Chemistry, Pharmaceutical Science, Biochemistry +13

Synthesis, Structure-Activity Relationships, and Pharmacological Evaluation of a Series of Fluorinated 3-Benzyl-5-Indolecarboxamides: Identification of 4-[[5-[((2R)-2-Methyl-4,4,4-trifluorobutyl)carbamoyl]-1-methylindol-3-yl]methyl]-3methoxy-N-[(2-methylphenyl)sulfonyl]benzamide, a Potent, Orally Active Antagonist of Leukotrienes D4 and E4

Robert T. Jacobs, Peter R Bernstein, Laura A. Cronk et al. · Journal of Medicinal Chemistry · 1994 · 41 citations · Full text

Synthesis and in vitro LTD4 antagonist activity of bicyclic and monocyclic cyclopentylurethane and cyclopentylacetamide N-arylsulfonyl amides

Victor G. Matassa, F.J. Brown, Peter R Bernstein et al. · Journal of Medicinal Chemistry · 1990 · 24 citations

Medicinal Chemistry, N-arylsulfonyl Amides, Heterocyclic +15