Design, Synthesis and Evaluation of d-Homophenylalanyl Epoxysuccinate Inhibitors of the Trypanosomal Cysteine Protease Cruzain

On the size of the active site in proteases. I. Papain

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Vinyl Sulfones as Mechanism-Based Cysteine Protease Inhibitors

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New convenient reagent for peptide syntheses

B. Belleau, G Mälek · Journal of the American Chemical Society · 1968 · 411 citations

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Cysteine Protease Inhibitors Cure an Experimental <i>Trypanosoma cruzi</i> Infection

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A malarial cysteine proteinase is necessary for hemoglobin degradation by Plasmodium falciparum.

Philip J. Rosenthal, James H. McKerrow, M Aikawa et al. · Journal of Clinical Investigation · 1988 · 328 citations · Full text

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