Concepedia

A public-private partnership to unlock the untargeted kinome

Stefan Knapp, Paulo Arruda, Julian Blagg, S.K. Burley, David H. Drewry, A.M. Edwards, Doriano Fabbro, Paul Gillespie, Nathanael S. Gray, Bernhard Küster,

Nature Chemical Biology · 2012 · 151 citations · 21 references

DOI

Concepts

References

21

Comprehensive analysis of kinase inhibitor selectivity

Mindy I. Davis, Jeremy P. Hunt, Sanna Herrgård et al. · Nature Biotechnology · 2011 · 2.4K citations · Full text

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Quantitative chemical proteomics reveals mechanisms of action of clinical ABL kinase inhibitors

Marcus Bantscheff, Dirk Eberhard, Yann Abraham et al. · Nature Biotechnology · 2007 · 1K citations

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Targeting Bcr–Abl by combining allosteric with ATP-binding-site inhibitors

Jianming Zhang, Francisco Adrián, Wolfgang Jahnke et al. · Nature · 2010 · 599 citations

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Characterization of a selective inhibitor of the Parkinson's disease kinase LRRK2

Xianming Deng, Nicolas Dzamko, Alan R. Prescott et al. · Nature Chemical Biology · 2011 · 431 citations · Full text

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Too many roads not taken

A.M. Edwards, Ruth Isserlin, Gary D. Bader et al. · Nature · 2011 · 431 citations · Full text

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