Bioorganic & Medicinal Chemistry Letters · 2011 · 14 citations · 13 references
PharmacyMedicinal ChemistryPharmacologyDrug DesignDrug DiscoveryStructure-activity RelationshipsChemical Space ExplorationDrug-target Interaction MappingHit-to-lead OptimizationLigand BindingPotency OptimizationSelectivity OptimizationCannabinoid AgonistsCannabinoid Receptor PharmacologyCompound Potency OptimizationHit-to-probe OptimizationOptimization Of Drug-like PropertiesProperty-based Drug DesignReceptor Binding OptimizationSelectivity Profile Optimization
13
Molecular characterization of a peripheral receptor for cannabinoids
Sean Munro, Kerrie L. Thomas, Muna Abu-Shaar · Nature · 1993 · 5.1K citations
Determination and characterization of a cannabinoid receptor in rat brain.
William A. Devane, F A Dysarz, M R Johnson et al. · Molecular Pharmacology · 1988 · 2.4K citations
Medicine, Neuroscience, Pharmacology +12
Cannabinoid receptor localization in brain.
Miles Herkenham, A B Lynn, M.D. Little et al. · Proceedings of the National Academy of Sciences · 1990 · 2.3K citations