Heather Grbic

Discovery of potent and selective PKC-θ inhibitors

Charles L. Cywin, Georg Dahmann, Anthony S. Prokopowicz et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 70 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

1,4-Diazepane compounds as potent and selective CB2 agonists: Optimization of metabolic stability

Doris Riether, Lifen Wu, Pier F. Cirillo et al. · Bioorganic & Medicinal Chemistry Letters · 2011 · 21 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

Automatable Formats of Higher Throughput ADMET Profiling for Drug Discovery Support

Paul V. Kaplita, Han-Bo Hu, Lisa Liu et al. · JALA Journal of the Association for Laboratory Automation · 2005 · 15 citations

Pharmacy, Medicinal Chemistry, Pharmacology +14

Aryl 1,4-diazepane compounds as potent and selective CB2 agonists: Optimization of drug-like properties and target independent parameters

Renée Zindell, Edward R. Walker, John Scott et al. · Bioorganic & Medicinal Chemistry Letters · 2011 · 14 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17