Anthony S. Prokopowicz

Three Mechanistically Distinct Kinase Assays Compared: Measurement of Intrinsic ATPase Activity Identified the Most Comprehensive Set of ITK Inhibitors

Mohammed A. Kashem, Richard M. Nelson, Jeffrey D. Yingling et al. · SLAS DISCOVERY · 2006 · 132 citations · Full text

Discovery of potent and selective PKC-θ inhibitors

Charles L. Cywin, Georg Dahmann, Anthony S. Prokopowicz et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 69 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Drug Target +7

Hit to Lead Account of the Discovery of a New Class of Inhibitors of Pim Kinases and Crystallographic Studies Revealing an Unusual Kinase Binding Mode

Kevin Qian, Lian Wang, Charles L. Cywin et al. · Journal of Medicinal Chemistry · 2009 · 69 citations · Full text

Pim Kinases, Pim-2 Sar, Molecular Biology +18

Evolution of the Thienopyridine Class of Inhibitors of IκB Kinase-β:  Part I:  Hit-to-Lead Strategies

Tina M. Morwick, Angela Berry, Janice R. Brickwood et al. · Journal of Medicinal Chemistry · 2006 · 67 citations · Full text

Discovery of 2-Phenylamino-imidazo[4,5-<i>h</i>]isoquinolin-9-ones:  A New Class of Inhibitors of Lck Kinase

Roger J. Snow, Mario Cardozo, Tina M. Morwick et al. · Journal of Medicinal Chemistry · 2002 · 63 citations · Full text