Paul V. Kaplita

Identification of pharmacological inhibitors of the MEK5/ERK5 pathway

Revati J. Tatake, Margaret M. O’Neill, Charles A. Kennedy et al. · Biochemical and Biophysical Research Communications · 2008 · 154 citations

Medicine, Receptor Tyrosine Kinase, Mechanism Of Action +4

γ-Aminobutyric acid action in guinea-pig ileal myenteric plexus

Paul V. Kaplita, Donald H. Waters, David J. Triggle · European Journal of Pharmacology · 1982 · 113 citations

Animal Physiology, γ-Aminobutyric Acid Action, Gastrointestinal Pharmacology +7

Tyrosine kinase assays adapted to homogeneous time-resolved fluorescence

Alfred J. Kolb, Paul V. Kaplita, Dave J. Hayes et al. · Drug Discovery Today · 1998 · 78 citations

Single Molecule Biophysics, Signal Transduction, Natural Sciences +8

Discovery of potent and selective PKC-θ inhibitors

Charles L. Cywin, Georg Dahmann, Anthony S. Prokopowicz et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 69 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Drug Target +7

Evolution of the Thienopyridine Class of Inhibitors of IκB Kinase-β:  Part I:  Hit-to-Lead Strategies

Tina M. Morwick, Angela Berry, Janice R. Brickwood et al. · Journal of Medicinal Chemistry · 2006 · 67 citations · Full text