Bioorganic & Medicinal Chemistry Letters · 2007 · 13 citations · 10 references
PharmacyMedicinal ChemistryPharmacologyDrug DesignHepatic PharmacokineticsMetabolic StabilityHepatic Drug MetabolismHepatic MetabolismHepatocyte StabilityLiver DiseaseMetabolic Stability OptimizationMicrosomal StabilityCytochrome P450 Human Liver MicrosomesHepatic Microsomal MetabolismHepatocyte Stability AssaysHigh-throughput Microsomal Stability ScreeningLiver Microsomal MetabolismMicrosomal Intrinsic ClearanceRat Liver Microsomes
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Katherine E. Cole, Christine A. Strick, Timothy Paradis et al. · The Journal of Experimental Medicine · 1998 · 879 citations · Full text
The prediction of human clearance from hepatic microsomal metabolism data.
Blockade of chemokine signaling in patients with multiple sclerosis
Frauke Zipp, HP Hartung, Jan Hillert et al. · Neurology · 2006 · 83 citations