An efficient synthesis for a new class antimalarial agent, 7-(2-carboxyethyl)-1,3-dihydro-1-hydroxy-2,1-benzoxaborole

An Antifungal Agent Inhibits an Aminoacyl-tRNA Synthetase by Trapping tRNA in the Editing Site

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Life Sciences, Biochemistry, Medicinal Chemistry +17

Discovery and structure–activity study of a novel benzoxaborole anti-inflammatory agent (AN2728) for the potential topical treatment of psoriasis and atopic dermatitis

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Pharmacy, Medicinal Chemistry, Pharmacology +17

Malaria's Drug Miracle in Danger

Martin Enserink · Science · 2010 · 116 citations

Veterinary Medicine, Infectious Diseases, Pharmacology +5

Synthesis and structure–activity relationships of novel benzoxaboroles as a new class of antimalarial agents

Yong-Kang Zhang, Jacob J. Plattner, Yvonne R. Freund et al. · Bioorganic & Medicinal Chemistry Letters · 2010 · 80 citations

Pharmacy, Medicinal Chemistry, Pharmacology +15

Design and synthesis of boron-containing PDE4 inhibitors using soft-drug strategy for potential dermatologic anti-inflammatory application

Yongkang Zhang, Jacob J. Plattner, Tsutomu Akama et al. · Bioorganic & Medicinal Chemistry Letters · 2010 · 41 citations

Pharmacy, Medicinal Chemistry, Pharmacology +13