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Further insights into the SAR of α-substituted cyclopropylamine derivatives as inhibitors of histone demethylase KDM1A

Marco Pieroni, Giannamaria Annunziato, Elisa Azzali, Paola Dessanti, Ciro Mercurio, Giuseppe Meroni, Paolo Trifiró, Paola Vianello, Manuela Villa, Claudia Beato,

European Journal of Medicinal Chemistry · 2015 · 31 citations · 26 references

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26

The protein data bank: A computer-based archival file for macromolecular structures

F. C. Bernstein, Thomas F. Koetzle, G. J. B. Williams et al. · Journal of Molecular Biology · 1977 · 8.6K citations

, , +13

Histone Demethylation Mediated by the Nuclear Amine Oxidase Homolog LSD1

Yujiang Geno Shi · Cell · 2004 · 3.9K citations · Full text

, , +8

Hypomethylation distinguishes genes of some human cancers from their normal counterparts

Andrew P. Feinberg, Bert Vogelstein · Nature · 1983 · 2.4K citations

, , +11

LSD1 demethylates repressive histone marks to promote androgen-receptor-dependent transcription

Eric Metzger, Melanie Wissmann, Na Yin et al. · Nature · 2005 · 1.7K citations

, , +11

New Model for Calculation of Solvation Free Energies:  Correction of Self-Consistent Reaction Field Continuum Dielectric Theory for Short-Range Hydrogen-Bonding Effects

Bryan Marten, Kyungsun Kim, Christian M. Cortis et al. · The Journal of Physical Chemistry · 1996 · 953 citations

, , +22