Concepedia

Ring contraction and rearrangement of 4-thiofuranose derivatives observed during DAST fluorination in the synthesis of l-2′-“up”-fluoro-4′-thiothymidine

Lak Shin Jeong, Hyung Ryong Moon, Su Jeong Yoo, Sun Nan Lee, Moon Woo Chun, Yoongho Lim

Tetrahedron Letters · 1998 · 29 citations · 6 references

DOI

Concepts

References

6

Activities of the four optical isomers of 2',3'-dideoxy-3'-thiacytidine (BCH-189) against human immunodeficiency virus type 1 in human lymphocytes

Raymond F. Schinazi, C. K. CHU, A Peck et al. · Antimicrobial Agents and Chemotherapy · 1992 · 265 citations · Full text

, , +9

Synthesis of enantiomerically pure (2'R,5'S)-(-)-1-(2-hydroxymethyloxathiolan-5-yl)cytosine as a potent antiviral agent against hepatitis B virus (HBV) and human immunodeficiency virus (HIV)

Joseph Warren Beach, Lak Shin Jeong, Antônio J. Alves et al. · The Journal of Organic Chemistry · 1992 · 192 citations

, , +6

Structure−Activity Relationships of 1-(2-Deoxy-2-fluoro-β-<scp>l</scp>-arabino- furanosyl)pyrimidine Nucleosides as Anti-Hepatitis B Virus Agents

Tianwei Ma, S. Balakrishna Pai, Yong Zhu et al. · Journal of Medicinal Chemistry · 1996 · 141 citations

, , +15

A Novel Synthesis of 2‘-Modified 2‘-Deoxy-4‘-thiocytidines from <scp>d</scp>-Glucose<sup>1</sup>

Yuichi Yoshimura, Kenji Kitano, Kohei Yamada et al. · The Journal of Organic Chemistry · 1997 · 101 citations

, , +13

Unanticipated retention of configuration in the DAST fluorination of deoxy-4′-thiopyrimidine nucleosides with “up” hydroxyl groups

Lak Shin Jeong, Marc C. Nicklaus, Cliff George et al. · Tetrahedron Letters · 1994 · 37 citations

, , +7