Concepedia
Journal of Fluorine Chemistry · 2008 · 16 citations · 10 references
BiochemistryNatural SciencesSingle Fluorine AtomDramatic EffectFluorous SynthesisOrganic ChemistryPeptide ScienceKey Aza-michael ReactionPeptide SynthesisChemistry
10
Peptidomimetics—Tailored Enzyme Inhibitors
Joachim Gante · Angewandte Chemie International Edition in English · 1994 · 814 citations
Peptide Engineering, Peptide Science, Pharmacotherapy +21
Trifluoroethylamines as amide isosteres in inhibitors of cathepsin K
W. Cameron Black, Christopher I. Bayly, Dana Davis et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 137 citations
Medicinal Chemistry, Derivative (Chemistry), Biochemistry +8
Difluoroethylamines as an amide isostere in inhibitors of cathepsin K
Élise Isabel, Christophe Mellon, Michael J. Boyd et al. · Bioorganic & Medicinal Chemistry Letters · 2010 · 111 citations · Full text
Medicinal Chemistry, Pharmaceutical Chemistry, Pharmaceutical Science +10
Identification of a potent and selective non-basic cathepsin K inhibitor
Chun Sing Li, Denis Deschênes, Sylvie Desmarais et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 87 citations · Full text
Biochemistry, Medicine, Natural Sciences +7
Synthesis, Structure and Conformation of Partially‐Modified Retro‐ and Retro‐Inverso ψ[NHCH(CF<sub>3</sub>)]Gly Peptides
Alessandro Volonterio, Stefano Bellosta, F. Bravin et al. · Chemistry - A European Journal · 2003 · 73 citations
Partially‐modified Retro‐, Engineering, Biochemistry +15