Teruki Hamada

Discovery of a Novel Pyrrole Derivative 1-[5-(2-Fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1<i>H</i>-pyrrol-3-yl]-<i>N</i>-methylmethanamine Fumarate (TAK-438) as a Potassium-Competitive Acid Blocker (P-CAB)

Yasuyoshi Arikawa, Haruyuki Nishida, Osamu Kurasawa et al. · Journal of Medicinal Chemistry · 2012 · 157 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17

Discovery of the First Potent and Orally Available Agonist of the Orphan G-Protein-Coupled Receptor 52

Masaki Setoh, Naoki Ishii, Mitsunori Kono et al. · Journal of Medicinal Chemistry · 2014 · 58 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Direct Drug Delivery of Low-Permeable Compounds to the Central Nervous System Via Intranasal Administration in Rats and Monkeys

Shinji Iwasaki, S. Yamamoto, Noriyasu Sano et al. · Pharmaceutical Research · 2019 · 37 citations

Pharmacy, Pharmaceutics, Pharmacology +13

Design and synthesis of 1-(1-benzothiophen-7-yl)-1H-pyrazole, a novel series of G protein-coupled receptor 52 (GPR52) agonists

Takashi Nakahata, Kazuyuki Tokumaru, Y. ITO et al. · Bioorganic & Medicinal Chemistry · 2018 · 33 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

Design and Identification of a GPR40 Full Agonist (<b>SCO-267</b>) Possessing a 2-Carbamoylphenyl Piperidine Moiety

Hideki Furukawa, Yasufumi Miyamoto, Yasuhiro Hirata et al. · Journal of Medicinal Chemistry · 2020 · 30 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17