Brian A. Chauder

Discovery of Potent Myeloid Cell Leukemia 1 (Mcl-1) Inhibitors Using Fragment-Based Methods and Structure-Based Design

Anders Friberg, Dominico Vigil, Bin Zhao et al. · Journal of Medicinal Chemistry · 2012 · 302 citations · Full text

Lead Compounds, Drug Target, Large Fragment Library +16

High-Throughput Screening Reveals a Small-Molecule Inhibitor of the Renal Outer Medullary Potassium Channel and Kir7.1

L. Michelle Lewis, Gautam Bhave, Brian A. Chauder et al. · Molecular Pharmacology · 2009 · 93 citations · Full text

Investigating Metabotropic Glutamate Receptor 5 Allosteric Modulator Cooperativity, Affinity, and Agonism: Enriching Structure-Function Studies and Structure-Activity Relationships

Karen J. Gregory, Meredith J. Noetzel, Jerri M. Rook et al. · Molecular Pharmacology · 2012 · 92 citations · Full text

Development of a Selective Small-Molecule Inhibitor of Kir1.1, the Renal Outer Medullary Potassium Channel

Gautam Bhave, Brian A. Chauder, Wen Liu et al. · Molecular Pharmacology · 2010 · 85 citations · Full text

Fragment-Based Screening of the Bromodomain of ATAD2

Mary J. Harner, Brian A. Chauder, Jason Phan et al. · Journal of Medicinal Chemistry · 2014 · 82 citations · Full text

Fragment Screen, Molecular Characterization, Fragment Hits +12