Michael J. Castaldi

Evaluation of Kilogram-Scale Sonagashira, Suzuki, and Heck Coupling Routes to Oncology Candidate CP-724,714

David H. Brown Ripin, Dennis E. Bourassa, Thomas A. Brandt et al. · Organic Process Research & Development · 2005 · 75 citations

Surgical Oncology, Engineering, Kilogram-scale Sonagashira +18

An Efficient and Cost-Effective Synthesis of 2-Phenyl-3-aminopyridine

Stéphane Caron, Steve S. Massett, David E. Bogle et al. · Organic Process Research & Development · 2001 · 43 citations

Combinatorial Chemistry, Key Intermediate, Engineering +11

In vitro activity of CP-99,219, a novel 7-(3-azabicyclo[3.1.0]hexyl) naphthyridone antimicrobial

Thomas D. Gootz, Katherine E. Brighty, Marge R. Anderson et al. · Diagnostic Microbiology and Infectious Disease · 1994 · 41 citations

Antimicrobial Drug Discovery, Biochemistry, Antibiotics +9

Synthesis of (1α,5α,6α)-6-Amino-3-azabicyclo[3.1.0]hexane, a Novel Achiral Diamine

Katherine E. Brighty, Michael J. Castaldi · Synlett · 2000 · 38 citations

Heterocyclic, Modified Curtius Rearrangement, Natural Sciences +9

3-Quinolinecarboxamides. A series of novel orally-active antiherpetic agents

Mark P. Wentland, Robert B. Perni, Peter H. Dorff et al. · Journal of Medicinal Chemistry · 1993 · 35 citations

Molecular Pharmacology, Medicinal Chemistry, Medicine +15