G. Toth

Design of an orally efficacious hydroxyethylamine (HEA) BACE-1 inhibitor in a preclinical animal model

Anh P. Truong, G. Toth, Gary D. Probst et al. · Bioorganic & Medicinal Chemistry Letters · 2010 · 48 citations · Full text

Pharmacological Study, Biochemistry, Medicine +9

Highly selective c-Jun N-terminal kinase (JNK) 2 and 3 inhibitors with in vitro CNS-like pharmacokinetic properties prevent neurodegeneration

Gary D. Probst, Simeon Bowers, Jennifer M. Sealy et al. · Bioorganic & Medicinal Chemistry Letters · 2010 · 44 citations · Full text

Medicine, Cell Death, Neuropharmacology +8

Design and synthesis of a novel, orally active, brain penetrant, tri-substituted thiophene based JNK inhibitor

Simeon Bowers, Anh P. Truong, R. Jeffrey Neitz et al. · Bioorganic & Medicinal Chemistry Letters · 2011 · 38 citations · Full text

Pharmaceutical Science, Tri-substituted Thiophene, Brain Penetrant +8

Improving the permeability of the hydroxyethylamine BACE-1 inhibitors: Structure–activity relationship of P2′ substituents

Anh P. Truong, Gary D. Probst, Jose Aquino et al. · Bioorganic & Medicinal Chemistry Letters · 2010 · 25 citations · Full text

Structure–activity Relationship, Molecular Pharmacology, Medicinal Chemistry +13

Characterization of degradation products of mometasone furoate.

Srikumar Sahasranaman, Manish Issar, G. Toth et al. · PubMed · 2004 · 11 citations

Asthma, Mometasone Furoate Degradation, Medicinal Chemistry +13