Katina Monzon

Discovery and Metabolic Stabilization of Potent and Selective 2-Amino-<i>N</i>-(adamant-2-yl) Acetamide 11β-Hydroxysteroid Dehydrogenase Type 1 Inhibitors

Jeffrey J. Rohde, Marina Pliushchev, Bryan K. Sorensen et al. · Journal of Medicinal Chemistry · 2006 · 76 citations · Full text

Medicinal Chemistry, Pharmacological Study, Biochemistry +11

Adamantane sulfone and sulfonamide 11-β-HSD1 Inhibitors

Bryan K. Sorensen, Martin Winn, Jeff Rohde et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 64 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Adamantane Sulfone +8

Discovery of adamantane ethers as inhibitors of 11β-HSD-1: Synthesis and biological evaluation

Jyoti Patel, Shuai Qi, Jürgen Dinges et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 41 citations · Full text

Medicinal Chemistry, Bioorganic Chemistry, Biochemistry +11

Adamantane 11-β-HSD-1 inhibitors: Application of an isocyanide multicomponent reaction

Bryan K. Sorensen, Jeff Rohde, Jiahong Wang et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 37 citations · Full text

Medicinal Chemistry, Medicine, Isocyanide Multicomponent Reaction +3

Synthesis and structural activity relationship of 11β-HSD1 inhibitors with novel adamantane replacements

Vince S. C. Yeh, Ravi Kurukulasuriya, David J. Madar et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 31 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Biochemistry +12