Robert E. Kyne

Rational Targeting of Active-Site Tyrosine Residues Using Sulfonyl Fluoride Probes

Erik C. Hett, Hua Xu, Kieran F. Geoghegan et al. · ACS Chemical Biology · 2015 · 191 citations

Molecular Pharmacology, Drug Target, Biochemistry +15

Enantioselective Construction of All-Carbon Quaternary Centers by Branch-Selective Pd-Catalyzed Allyl–Allyl Cross-Coupling

Ping Zhang, Hai Le, Robert E. Kyne et al. · Journal of the American Chemical Society · 2011 · 179 citations

Covalent Enzyme Inhibition through Fluorosulfate Modification of a Noncatalytic Serine Residue

Olugbeminiyi Fadeyi, Lise R. Hoth, Chulho Choi et al. · ACS Chemical Biology · 2017 · 134 citations

Drug Target, Bioorganic Chemistry, Molecular Biology +22

Synthesis of Pyrazoles from 1,3-Diols via Hydrogen Transfer Catalysis

Daniel C. Schmitt, Alexandria P. Taylor, Andrew C. Flick et al. · Organic Letters · 2015 · 62 citations

1,3-Diols Engage, Engineering, 1,4-Disubstituted Pyrazoles +8

Chemoselective Preparation of Clickable Aryl Sulfonyl Fluoride Monomers: A Toolbox of Highly Functionalized Intermediates for Chemical Biology Probe Synthesis

Olugbeminiyi Fadeyi, Mihir D. Parikh, Ming Z. Chen et al. · ChemBioChem · 2016 · 55 citations