Mihir D. Parikh

Rational Targeting of Active-Site Tyrosine Residues Using Sulfonyl Fluoride Probes

Erik C. Hett, Hua Xu, Kieran F. Geoghegan et al. · ACS Chemical Biology · 2015 · 191 citations

Molecular Pharmacology, Drug Target, Biochemistry +15

Identification of <i>N</i>-{<i>cis</i>-3-[Methyl(7<i>H</i>-pyrrolo[2,3-<i>d</i>]pyrimidin-4-yl)amino]cyclobutyl}propane-1-sulfonamide (PF-04965842): A Selective JAK1 Clinical Candidate for the Treatment of Autoimmune Diseases

Michael L. Vazquez, Neelu Kaila, Joseph W. Strohbach et al. · Journal of Medicinal Chemistry · 2018 · 160 citations · Full text

Immunodeficiencies, Janus Kinases, Immunology +22

Identification of a Chemical Probe for Family VIII Bromodomains through Optimization of a Fragment Hit

Brian S. Gerstenberger, John D. Trzupek, C. Tallant et al. · Journal of Medicinal Chemistry · 2016 · 107 citations · Full text

Molecular Biology, Chemical Biology, Pharmaceutical Chemistry +22

Chemoselective Preparation of Clickable Aryl Sulfonyl Fluoride Monomers: A Toolbox of Highly Functionalized Intermediates for Chemical Biology Probe Synthesis

Olugbeminiyi Fadeyi, Mihir D. Parikh, Ming Z. Chen et al. · ChemBioChem · 2016 · 55 citations

Porphyrins with exocyclic rings. Part 19: Efficient syntheses of phenanthrolinoporphyrins

Timothy D. Lash, Yanning Lin, Bennett H. Novak et al. · Tetrahedron · 2005 · 49 citations

Engineering, Organic Chemistry, Exocyclic Rings +5