Michael L. Vazquez

Identification of <i>N</i>-{<i>cis</i>-3-[Methyl(7<i>H</i>-pyrrolo[2,3-<i>d</i>]pyrimidin-4-yl)amino]cyclobutyl}propane-1-sulfonamide (PF-04965842): A Selective JAK1 Clinical Candidate for the Treatment of Autoimmune Diseases

Michael L. Vazquez, Neelu Kaila, Joseph W. Strohbach et al. · Journal of Medicinal Chemistry · 2018 · 160 citations · Full text

Immunodeficiencies, Janus Kinases, Immunology +22

Synthesis, Crystal Structure, and Activity of Pyrazole-Based Inhibitors of p38 Kinase

Matthew J. Graneto, Ravi G. Kurumbail, Michael L. Vazquez et al. · Journal of Medicinal Chemistry · 2007 · 64 citations · Full text

Distinction of microsomal prostaglandin E synthase-1 (mPGES-1) inhibition from cyclooxygenase-2 inhibition in cells using a novel, selective mPGES-1 inhibitor

Gabriel Mbalaviele, Adele M. Pauley, Alexander F. Shaffer et al. · Biochemical Pharmacology · 2010 · 64 citations

Selective Mpges-1 Inhibitor, Biochemistry, Medicine +8

Selective inducible microsomal prostaglandin E2 synthase-1 (mPGES-1) inhibitors derived from an oxicam template

Jane Wang, David C. Limburg, Jeff Carter et al. · Bioorganic & Medicinal Chemistry Letters · 2010 · 61 citations · Full text

Medicinal Chemistry, Biochemistry, Oxicam Template +9

Inhibitors of HIV-1 Protease Containing the Novel and Potent (R)-(Hydroxyethyl)sulfonamide Isostere

Michael L. Vazquez, Martin L. Bryant, Michael Clare et al. · Journal of Medicinal Chemistry · 1995 · 48 citations · Full text

Altmetric Attention Score, Antiviral Drug, Chemical Biology +16