Yasunori Kawakita

(1<i>S</i>)-1,5-Anhydro-1-[5-(4-ethoxybenzyl)-2-methoxy-4-methylphenyl]-1-thio-<scp>d</scp>-glucitol (TS-071) is a Potent, Selective Sodium-Dependent Glucose Cotransporter 2 (SGLT2) Inhibitor for Type 2 Diabetes Treatment

Hiroyuki Kakinuma, Takahiro Oi, Yuko Hashimoto-Tsuchiya et al. · Journal of Medicinal Chemistry · 2010 · 158 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Increase of Intracellular Glutathione by Low-Dose .GAMMA.-Ray Irradiation Is Mediated by Transcription Factor AP-1 in RAW 264.7 Cells.

Yasunori Kawakita, Masahiko Ikekita, Risa Kurozumi et al. · Biological and Pharmaceutical Bulletin · 2003 · 42 citations · Full text

Medicine, Molecular Biology, Radiation Biophysics +14

Efficacy of a glycine transporter 1 inhibitor TASP0315003 in animal models of cognitive dysfunction and negative symptoms of schizophrenia

Shigeyuki Chaki, Toshiharu Shimazaki, Jun-ichi Karasawa et al. · Psychopharmacology · 2015 · 27 citations

Medicine, Neuroscience, Pharmacology +17

Synthesis, in vitro pharmacology, and pharmacokinetic profiles of 2-[1-amino-1-carboxy-2-(9H-xanthen-9-yl)-ethyl]-1-fluorocyclopropanecarboxylic acid and its 6-heptyl ester, a potent mGluR2 antagonist

Kazunari Sakagami, Akito Yasuhara, Shigeyuki Chaki et al. · Bioorganic & Medicinal Chemistry · 2008 · 20 citations · Full text

Pharmacy, Pharmacokinetics, Pharmacology +6

IN VITRO AND IN VIVO EVALUATION OF THE METABOLISM AND BIOAVAILABILITY OF ESTER PRODRUGS OF MGS0039 (3-(3,4-DICHLOROBENZYLOXY)-2-AMINO-6-FLUOROBICYCLO[3.1.0]HEXANE-2,6-DICARBOXYLIC ACID), A POTENT METABOTROPIC GLUTAMATE RECEPTOR ANTAGONIST

Masato Nakamura, Yasunori Kawakita, Akito Yasuhara et al. · Drug Metabolism and Disposition · 2005 · 14 citations

Pharmacy, Pharmacokinetics, Pharmacology +16