Craig A. Stump

Mechanism based neurotoxicity of mGlu5 positive allosteric modulators – Development challenges for a promising novel antipsychotic target

Sophie Parmentier‐Batteur, Peter H. Hutson, Karsten Menzel et al. · Neuropharmacology · 2013 · 93 citations

Molecular Pharmacology, Molecular Neuroscience, Development Challenges +11

Discovery of MK-3207: A Highly Potent, Orally Bioavailable CGRP Receptor Antagonist

Ian M. Bell, Steven N. Gallicchio, Michael R. Wood et al. · ACS Medicinal Chemistry Letters · 2010 · 63 citations

Non-peptide calcitonin gene-related peptide receptor antagonists from a benzodiazepinone lead

Theresa M. Williams, Craig A. Stump, Diem N. Nguyen et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 52 citations · Full text

Biochemistry, Medicine, Receptor (Biochemistry) +7

Benzodiazepine calcitonin gene-related peptide (CGRP) receptor antagonists: Optimization of the 4-substituted piperidine

Christopher S. Burgey, Craig A. Stump, Diem N. Nguyen et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 51 citations · Full text

Biochemistry, Functional Selectivity, Medicine +8

Structural characterization of nonactive site, TrkA-selective kinase inhibitors

Hua-Poo Su, Keith Rickert, Christine Burlein et al. · Proceedings of the National Academy of Sciences · 2016 · 48 citations · Full text

Nonactive Site, Medicinal Chemistry, Drug Target +15