Concepedia

Non-peptide calcitonin gene-related peptide receptor antagonists from a benzodiazepinone lead

Theresa M. Williams, Craig A. Stump, Diem N. Nguyen, Amy G. Quigley, Ian M. Bell, Steven N. Gallicchio, C. Blair Zartman, Bang-Lin Wan, Kimberly Della Penna, Priya Kunapuli,

Bioorganic & Medicinal Chemistry Letters · 2006 · 52 citations · 15 references

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References

15

Calcitonin gene-related peptide is a potent vasodilator

Susan D. Brain, T.J. Williams, John R. Tippins et al. · Nature · 1985 · 2.1K citations

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Methods for drug discovery: development of potent, selective, orally effective cholecystokinin antagonists

B. Evans, Kenneth E. Rittle, Mark G. Bock et al. · Journal of Medicinal Chemistry · 1988 · 1.4K citations · Full text

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Calcitonin Gene–Related Peptide Receptor Antagonist BIBN 4096 BS for the Acute Treatment of Migraine

Jes Olesen, Hans‐Christoph Diener, Ingo W. Husstedt et al. · New England Journal of Medicine · 2004 · 1.2K citations · Full text

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Migraine Diagnosis and Treatment: Results From the American Migraine Study II

Richard B. Lipton, Seymour Diamond, Michael L. Reed et al. · Headache The Journal of Head and Face Pain · 2001 · 729 citations

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Receptor Activity-modifying Protein 1 Determines the Species Selectivity of Non-peptide CGRP Receptor Antagonists

John Mallee, Christopher Salvatore, Beatrice LeBourdellès et al. · Journal of Biological Chemistry · 2002 · 191 citations · Full text

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