Susan Lockhead

Synthesis and Structure−Activity Relationship of Novel 6-Aryl-1,4- dihydrobenzo[<i>d</i>][1,3]oxazine-2-thiones as Progesterone Receptor Modulators Leading to the Potent and Selective Nonsteroidal Progesterone Receptor Agonist Tanaproget

Andrew Fensome, Reinhold H. W. Bender, Rajiv Chopra et al. · Journal of Medicinal Chemistry · 2005 · 91 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Characterization of HKI-272 Covalent Binding to Human Serum Albumin

Jianyao Wang, Xiao Xian Li-Chan, Jim Atherton et al. · Drug Metabolism and Disposition · 2010 · 61 citations

Pharmacy, Biochemistry, Molecular Biology +16

(1-(4-(Naphthalen-2-yl)pyrimidin-2-yl)piperidin-4-yl)methanamine: A Wingless β-Catenin Agonist That Increases Bone Formation Rate

Jeffrey C. Pelletier, Joseph T. Lundquist, A. Gilbert et al. · Journal of Medicinal Chemistry · 2009 · 53 citations · Full text

Pharmacy, Pharmacokinetics, Pharmacology +15

Reversible Covalent Binding of Neratinib to Human Serum Albumin In Vitro

Appavu Chandrasekaran, Li Shen, Susan Lockhead et al. · Drug Metabolism Letters · 2010 · 39 citations

Medicine, Biochemistry, Pharmacology +15

5-(3-Cyclopentyl-2-thioxo-2,3-dihydro-1H-benzimidazol-5-yl)-1-methyl-1H-pyrrole-2-carbonitrile: A novel, highly potent, selective, and orally active non-steroidal progesterone receptor agonist

Puwen Zhang, Eugene A. Terefenko, Jeffrey C. Kern et al. · Bioorganic & Medicinal Chemistry · 2007 · 18 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +8