Eugene A. Terefenko

Potent nonsteroidal progesterone receptor agonists: Synthesis and SAR study of 6-aryl benzoxazines

Puwen Zhang, Eugene A. Terefenko, Andrew Fensome et al. · Bioorganic & Medicinal Chemistry Letters · 2002 · 117 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +11

6-Aryl-1,4-dihydro-benzo[<i>d</i>][1,3]oxazin- 2-ones:  A Novel Class of Potent, Selective, and Orally Active Nonsteroidal Progesterone Receptor Antagonists

Puwen Zhang, Eugene A. Terefenko, Andrew Fensome et al. · Journal of Medicinal Chemistry · 2002 · 106 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +13

Synthesis and Structure−Activity Relationship of Novel 6-Aryl-1,4- dihydrobenzo[<i>d</i>][1,3]oxazine-2-thiones as Progesterone Receptor Modulators Leading to the Potent and Selective Nonsteroidal Progesterone Receptor Agonist Tanaproget

Andrew Fensome, Reinhold H. W. Bender, Rajiv Chopra et al. · Journal of Medicinal Chemistry · 2005 · 91 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Novel 6-aryl-1,4-dihydrobenzo[d][1,3]oxazine-2-thiones as potent, selective, and orally active nonsteroidal progesterone receptor agonists

Puwen Zhang, Eugene A. Terefenko, Andrew Fensome et al. · Bioorganic & Medicinal Chemistry Letters · 2003 · 61 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +8

Thiourea inhibitors of herpes viruses. Part 2: N-Benzyl-N′-arylthiourea inhibitors of CMV

Jonathan D. Bloom, Russell G. Dushin, Kevin J. Curran et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 60 citations

Life Sciences, Medicinal Chemistry, Microbiology +6