Armelle Le Gall

1,3-Dimethyl Benzimidazolones Are Potent, Selective Inhibitors of the BRPF1 Bromodomain

Emmanuel H. Demont, Paul Bamborough, Chun‐wa Chung et al. · ACS Medicinal Chemistry Letters · 2014 · 91 citations · Full text

Life Sciences, Medicinal Chemistry, Molecular Biology +14

Age, religious beliefs, and sexual attitudes

Armelle Le Gall, Étienne Mullet, Sheila Rivière Shafighi · The Journal of Sex Research · 2002 · 82 citations

Social Sciences, Psychology, Social Psychology +7

The discovery and optimisation of pyrido[2,3-d]pyrimidine-2,4-diamines as potent and selective inhibitors of mTOR kinase

Karine Malagu, Heather M. E. Duggan, Keith Menear et al. · Bioorganic & Medicinal Chemistry Letters · 2009 · 80 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

Discovery of a Bromodomain and Extraterminal Inhibitor with a Low Predicted Human Dose through Synergistic Use of Encoded Library Technology and Fragment Screening

Christopher R. Wellaway, Dominique Amans, Paul Bamborough et al. · Journal of Medicinal Chemistry · 2020 · 71 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

GSK6853, a Chemical Probe for Inhibition of the BRPF1 Bromodomain

Paul Bamborough, Heather Barnett, Isabelle Becher et al. · ACS Medicinal Chemistry Letters · 2016 · 66 citations · Full text

Life Sciences, Medicinal Chemistry, Molecular Biology +14