Heather Barnett

GSK789: A Selective Inhibitor of the First Bromodomains (BD1) of the Bromo and Extra Terminal Domain (BET) Proteins

Robert J. Watson, Paul Bamborough, Heather Barnett et al. · Journal of Medicinal Chemistry · 2020 · 84 citations · Full text

Chemoprevention Strategy, Immunology, Molecular Biology +21

Structure-Based Optimization of Naphthyridones into Potent ATAD2 Bromodomain Inhibitors

Paul Bamborough, Chun‐wa Chung, Rebecca C. Furze et al. · Journal of Medicinal Chemistry · 2015 · 83 citations · Full text

Molecular Docking, Combinatorial Chemistry, Medicinal Chemistry +14

Discovery of a Bromodomain and Extraterminal Inhibitor with a Low Predicted Human Dose through Synergistic Use of Encoded Library Technology and Fragment Screening

Christopher R. Wellaway, Dominique Amans, Paul Bamborough et al. · Journal of Medicinal Chemistry · 2020 · 69 citations · Full text

Defining STEAM Approaches for Higher Education

Claudia Carter, Heather Barnett, Kathryn Burns et al. · European Journal of STEM Education · 2021 · 69 citations · Full text

Inclusive Steam Education, Stem Education, Steam Practices +14

GSK6853, a Chemical Probe for Inhibition of the BRPF1 Bromodomain

Paul Bamborough, Heather Barnett, Isabelle Becher et al. · ACS Medicinal Chemistry Letters · 2016 · 64 citations · Full text

Halogenation, Chromatin, Micromolar Activity +14