Tiffany Carpenter

Discovery of Highly Potent and Selective Small Molecule ADAMTS-5 Inhibitors That Inhibit Human Cartilage Degradation via Encoded Library Technology (ELT)

Hongfeng Deng, Heather P. O’Keefe, Christopher P. Davie et al. · Journal of Medicinal Chemistry · 2012 · 149 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +14

Discovery, Synthesis, and Biological Evaluation of Thiazoloquin(az)olin(on)es as Potent CD38 Inhibitors

Curt D. Haffner, J. David Becherer, Eric E. Boros et al. · Journal of Medicinal Chemistry · 2015 · 136 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13

Discovery of 4-Amino-8-quinoline Carboxamides as Novel, Submicromolar Inhibitors of NAD-Hydrolyzing Enzyme CD38

J. David Becherer, Eric E. Boros, Tiffany Carpenter et al. · Journal of Medicinal Chemistry · 2015 · 56 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

Genetic Ablation of CD38 Protects against Western Diet-Induced Exercise Intolerance and Metabolic Inflexibility

Shian-Huey Chiang, W. Wallace Harrington, Guizhen Luo et al. · PLoS ONE · 2015 · 44 citations · Full text

Life Sciences, Biochemistry, Physiology +17

Substituted N-{3-[(1,1-dioxido-1,2-benzothiazol-3-yl)(phenyl)amino]propyl}benzamide analogs as potent Kv1.3 ion channel blockers. Part 2

Curt D. Haffner, Stephen A. Thomson, Yu Guo et al. · Bioorganic & Medicinal Chemistry Letters · 2010 · 13 citations · Full text

Natural Sciences, Medicinal Chemistry, Pharmacology +11