Structure–Activity Relationship of Pyrrolyl Diketo Acid Derivatives as Dual Inhibitors of HIV-1 Integrase and Reverse Transcriptase Ribonuclease H Domain

Giuliana Cuzzucoli Crucitti, Mathieu Métifiot, Luca Pescatori, +14

Journal of Medicinal Chemistry

Structure–activity RelationshipHiv-1 IntegraseMolecular BiologyAntiviral DrugMedicinal Chemistry +16

Identification of Highly Conserved Residues Involved in Inhibition of HIV-1 RNase H Function by Diketo Acid Derivatives

Angela Corona, Francesco Saverio Di Leva, Sylvain Thierry, +11

Antimicrobial Agents and Chemotherapy

Chemical BiologyRnase HBiochemistryNatural SciencesHuman Retrovirus +13

Inhibition of <i>Leishmania infantum</i> trypanothione reductase by diaryl sulfide derivatives

Francesco Saccoliti, Gabriella Angiulli, Giovanni Pupo, +11

Journal of Enzyme Inhibition and Medicinal Chemistry

Monotopic and heteroditopic calix[4]arene receptors as hosts for pyridinium and viologen ion pairs: a solution and solid-state study

Luca Pescatori, Arturo Arduini, Andrea Pochini, +3

Organic & Biomolecular Chemistry

Dimethylviologen SaltsGuest Ion PairBiochemistryNatural SciencesBinding Efficiency +8

6-(1-Benzyl-1<i>H</i>-pyrrol-2-yl)-2,4-dioxo-5-hexenoic Acids as Dual Inhibitors of Recombinant HIV-1 Integrase and Ribonuclease H, Synthesized by a Parallel Synthesis Approach

Roberta Costi, Mathieu Métifiot, Francesca Esposito, +11

Journal of Medicinal Chemistry

Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV Integrase and their Activity against RNase H Function of Reverse Transcriptase

Roberta Costi, Mathieu Métifiot, Suhman Chung, +17

Journal of Medicinal Chemistry

Effects of polyphenol compounds on influenza A virus replication and definition of their mechanism of action

Rossella Fioravanti, Ignacio Celestino, Roberta Costi, +8

Bioorganic & Medicinal Chemistry

Viral ReplicationPolyphenol CompoundsMedicineVirologyInfluenza Vaccine +3

<i>N</i>-Substituted Quinolinonyl Diketo Acid Derivatives as HIV Integrase Strand Transfer Inhibitors and Their Activity against RNase H Function of Reverse Transcriptase

Luca Pescatori, Mathieu Métifiot, Suhman Chung, +17

Journal of Medicinal Chemistry

Ribonuclease HMolecular BiologyStrand TransferTheir ActivityAntiviral Drug +17

Discovery and Pharmacological Profile of New 1<i>H</i>-Indazole-3-carboxamide and 2<i>H</i>-Pyrrolo[3,4-<i>c</i>]quinoline Derivatives as Selective Serotonin 4 Receptor Ligands

Guido Furlotti, Maria Alessandra Alisi, Claudia Apicella, +15

Journal of Medicinal Chemistry

Molecular PharmacologyMedicinal ChemistryPharmacological StudyBiochemistryFunctional Selectivity +12

Salmonella enterica serovar Typhimurium growth is inhibited by the concomitant binding of Zn(II) and a pyrrolyl-hydroxamate to ZnuA, the soluble component of the ZnuABC transporter

Andrea Ilari, Luca Pescatori, Roberto Di Santo, +6

Biochimica et Biophysica Acta (BBA) - General Subjects

Medical MicrobiologyBiochemistryVirulence FactorPathogenesisSerovar Typhimurium Growth +8