Francesco Saverio Di Leva

Design, Synthesis, and Biological Evaluation of Potent Dual Agonists of Nuclear and Membrane Bile Acid Receptors

Claudio D’Amore, Francesco Saverio Di Leva, Valentina Sepe et al. · Journal of Medicinal Chemistry · 2014 · 93 citations · Full text

Medicinal Chemistry, Lipid Synthesis, Biochemistry +15

Rational Improvement of the Affinity and Selectivity of Integrin Binding of Grafted Lasso Peptides

Julian D. Hegemann, Mariarosaria De Simone, Marcel Zimmermann et al. · Journal of Medicinal Chemistry · 2014 · 92 citations · Full text

Engineering, Peptide Engineering, Molecular Biology +23

Modification on Ursodeoxycholic Acid (UDCA) Scaffold. Discovery of Bile Acid Derivatives As Selective Agonists of Cell-Surface G-Protein Coupled Bile Acid Receptor 1 (GP-BAR1)

Valentina Sepe, Barbara Renga, Carmen Festa et al. · Journal of Medicinal Chemistry · 2014 · 90 citations · Full text

Molecular Pharmacology, Molecular Physiology, Biochemistry +14

Mechanistic insight into ligand binding to G-quadruplex DNA

Francesco Saverio Di Leva, Ettore Novellino, Andrea Cavalli et al. · Nucleic Acids Research · 2014 · 86 citations · Full text

Stable Peptides Instead of Stapled Peptides: Highly Potent αvβ6‐Selective Integrin Ligands

Oleg V. Maltsev, Udaya Kiran Marelli, Tobias G. Kapp et al. · Angewandte Chemie International Edition · 2015 · 73 citations