2-Methyl-6-(phenylethynyl)-pyridine (MPEP), a potent, selective and systemically active mGlu5 receptor antagonist

F. Gasparini, Kurt Lingenhöhl, Natacha Stoehr, +15

Neuropharmacology

BiochemistryFunctional SelectivityMedicineMechanism Of ActionReceptor (Biochemistry) +5

5-Phosphonomethylquinoxalinediones as competitive NMDA receptor antagonists with a preference for the human 1A/2A, rather than 1A/2B receptor composition

Yves P. Auberson, Hans Allgeier, Serge Bischoff, +3

Bioorganic & Medicinal Chemistry Letters

BiochemistryFunctional SelectivityMedicineMechanism Of ActionReceptor (Biochemistry) +5

SIB-1757 and SIB-1893: Selective, Noncompetitive Antagonists of Metabotropic Glutamate Receptor Type 5

Mark A. Varney, Nicholas D. P. Cosford, Christine Jachec, +12

Journal of Pharmacology and Experimental Therapeutics

CGP 37849 and CGP 39551: novel and potent competitive N‐methyl‐<scp>d</scp>‐aspartate receptor antagonists with oral activity

Graham E. Fagg, H.‐R. Olpe, M.F. Pozza, +12

British Journal of Pharmacology

Molecular PharmacologyCgp 37849BiochemistryMedicineSynaptic Transmission +13

The competitive NMDA receptor antagonists CGP 37849 and CGP 39551 are potent, orally-active anticonvulsants in rodents

Markus Schmutz, Ch. Portet, A. Jeker, +7

Naunyn-Schmiedeberg s Archives of Pharmacology

NeurophysiologyMedicineNeurotransmitterNeuropharmacologyExperimental Pharmacology +9

ABP688, a novel selective and high affinity ligand for the labeling of mGlu5 receptors: Identification, in vitro pharmacology, pharmacokinetic and biodistribution studies

Samuel Hintermann, Ivo Vranesic, Hans Allgeier, +8

Bioorganic & Medicinal Chemistry

Mglu5 ReceptorsBiochemistryG Protein-coupled ReceptorMedicineFunctional Selectivity +7

Struktur der Pachybiose und Asclepobiose. Desoxyzucker, 44. Mitteilung

Hans Allgeier

Helvetica Chimica Acta

Unicellular OrganismBiosynthesisBioorganic ChemistryBiochemistryStruktur Der Pachybiose +13

Differentiation of Glycine Antagonist Sites ofN-Methyl-d-aspartate Receptor Subtypes

Michael Honer, Dietmar Benke, Bodo Laube, +8

Journal of Biological Chemistry

Molecular distinction of three N-methyl-D-aspartate-receptor subtypes in situ and developmental receptor maturation demonstrated with the photoaffinity ligand 125I-labeled CGP 55802A.

Thomas M. Marti, Dietmar Benke, S. Mertens, +7

Proceedings of the National Academy of Sciences

NeurotransmitterMolecular BiologyOptogeneticsDevelopmental Receptor MaturationMolecular Pharmacology +23

Die Glykoside der Wurzeln von <i>Kanahia laniflora</i> (F<scp>ORSSK</scp>.) R. B<scp>R</scp>. 1. Mitteilung: Isolierungen. Glykoside und Aglykone, 299. Mitteilung

B.M. Kapur, Hans Allgeier, T. Reichstein

Helvetica Chimica Acta