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5-Phosphonomethylquinoxalinediones as competitive NMDA receptor antagonists with a preference for the human 1A/2A, rather than 1A/2B receptor composition

Yves P. Auberson, Hans Allgeier, Serge Bischoff, Kurt Lingenhoehl, Robert Moretti, Markus Schmutz

Bioorganic & Medicinal Chemistry Letters · 2002 · 222 citations · 12 references

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12

The Binding of [<sup>3</sup>H]AMPA, a Structural Analogue of Glutamic Acid, to Rat Brain Membranes

Tage Honoré, Jørn Lauridsen, Povl Krogsgaard‐Larsen · Journal of Neurochemistry · 1982 · 228 citations

, , +17

CGS 19755, a selective and competitive N-methyl-D-aspartate-type excitatory amino acid receptor antagonist.

John Lehmann, A. Hutchison, Stephen E. McPherson et al. · Journal of Pharmacology and Experimental Therapeutics · 1988 · 226 citations

, , +17

[3H]CGP 39653: a new N-methyl-D-aspartate antagonist radioligand with low nanomolar affinity in rat brain

Matthew A. Sills, Graham E. Fagg, Mario F. Pozza et al. · European Journal of Pharmacology · 1991 · 211 citations

, , +12

The competitive NMDA receptor antagonists CGP 37849 and CGP 39551 are potent, orally-active anticonvulsants in rodents

Markus Schmutz, Ch. Portet, A. Jeker et al. · Naunyn-Schmiedeberg s Archives of Pharmacology · 1990 · 137 citations

, , +11

Synthesis of organophosphorus compounds via silyl esters of phosphorous acids

Kamyar Afarinkia, Charles W. Rees, J. I. G. Cadogan · Tetrahedron · 1990 · 95 citations

, , +6