Matteo Falsini

Design, Synthesis, and Pharmacological Characterization of 2-(2-Furanyl)thiazolo[5,4-<i>d</i>]pyrimidine-5,7-diamine Derivatives: New Highly Potent A_2AAdenosine Receptor Inverse Agonists with Antinociceptive Activity

Flavia Varano, Daniela Catarzi, Fabrizio Vincenzi et al. · Journal of Medicinal Chemistry · 2016 · 56 citations · Full text

Structural investigations on coumarins leading to chromeno[4,3-c]pyrazol-4-ones and pyrano[4,3-c]pyrazol-4-ones: New scaffolds for the design of the tumor-associated carbonic anhydrase isoforms IX and XII

Alessandro Bonardi, Matteo Falsini, Daniela Catarzi et al. · European Journal of Medicinal Chemistry · 2018 · 53 citations · Full text

Combinatorial Chemistry, Medicinal Chemistry, Biochemistry +6

Crystal Structure and Subsequent Ligand Design of a Nonriboside Partial Agonist Bound to the Adenosine A_2A Receptor

Tasia Amelia, Jacobus P. D. van Veldhoven, Matteo Falsini et al. · Journal of Medicinal Chemistry · 2021 · 40 citations · Full text

The 1,2,4-Triazolo[4,3-<i>a</i>]pyrazin-3-one as a Versatile Scaffold for the Design of Potent Adenosine Human Receptor Antagonists. Structural Investigations to Target the A_2AReceptor Subtype

Matteo Falsini, Lucia Squarcialupi, Daniela Catarzi et al. · Journal of Medicinal Chemistry · 2017 · 35 citations · Full text

The aminopyridine-3,5-dicarbonitrile core for the design of new non-nucleoside-like agonists of the human adenosine A2B receptor

Marco Betti, Daniela Catarzi, Flavia Varano et al. · European Journal of Medicinal Chemistry · 2018 · 34 citations · Full text

New Non-nucleoside-like Agonists, Biochemistry, Functional Selectivity +7