Jacobus P. D. van Veldhoven

Predicting Binding Affinities for GPCR Ligands Using Free-Energy Perturbation

Eelke B. Lenselink, Julien Louvel, Anna F. Forti et al. · ACS Omega · 2016 · 145 citations · Full text

False Positives in a Reporter Gene Assay: Identification and Synthesis of Substituted <i>N</i>-Pyridin-2-ylbenzamides as Competitive Inhibitors of Firefly Luciferase

Laura H. Heitman, Jacobus P. D. van Veldhoven, Annelien J.M. Zweemer et al. · Journal of Medicinal Chemistry · 2008 · 65 citations · Full text

Drug Target, Firefly Luciferase, Molecular Biology +20

Dual-Point Competition Association Assay: A Fast and High-Throughput Kinetic Screening Method for Assessing Ligand-Receptor Binding Kinetics

Dong Guo, Erika J.H. van Dorp, Thea Mulder‐Krieger et al. · SLAS DISCOVERY · 2012 · 65 citations · Full text

A Series of 2,4-Disubstituted Quinolines as a New Class of Allosteric Enhancers of the Adenosine A₃Receptor

Laura H. Heitman, Anikó Göblyös, Annelien J.M. Zweemer et al. · Journal of Medicinal Chemistry · 2009 · 62 citations · Full text

Binding Kinetics of ZM241385 Derivatives at the Human Adenosine A_2A Receptor

Dong Guo, Lizi Xia, Jacobus P. D. van Veldhoven et al. · ChemMedChem · 2014 · 49 citations