Jacobus P. D. van Veldhoven

Author

Leiden University

Also Known As

Jacobus P D van Veldhoven, Jacobus P. D. van Veldhoven, Jacobus P. D. van Veldhoven, Jacobus P.D. van Veldhoven

Publications

823

Citations

H-Index

Concepts

All Affiliations

Leiden University Centre for Human Drug Research Medical College of Wisconsin

About

Jacobus P. D. van Veldhoven is an author at Leiden University specializing in biochemistry, pharmacology, and medicine.

Top Concepts

#	Concept	H-Index	Publications	Citations
1	Biochemistry	6	6	190
2	Medicine	5	5	171
3	Natural Sciences	4	4	126
4	Chemical Biology	4	4	126
5	Chemistry	1	1	25

Jacobus P. D. van Veldhoven

Publications

783

Citations

H-Index

Page 1

	Year	Citations
Predicting Binding Affinities for GPCR Ligands Using Free-Energy Perturbation Eelke B. Lenselink, Julien Louvel, Anna F. Forti, ACS Omega	2016	145
False Positives in a Reporter Gene Assay: Identification and Synthesis of Substituted <i>N</i>-Pyridin-2-ylbenzamides as Competitive Inhibitors of Firefly Luciferase Laura H. Heitman, Jacobus P. D. van Veldhoven, Annelien J.M. Zweemer, Journal of Medicinal Chemistry Drug TargetFirefly LuciferaseMolecular BiologyLuciferase Reporter-gene AssaysChemical Biology	2008	65
Dual-Point Competition Association Assay: A Fast and High-Throughput Kinetic Screening Method for Assessing Ligand-Receptor Binding Kinetics Dong Guo, Erika J.H. van Dorp, Thea Mulder‐Krieger, SLAS DISCOVERY	2012	65
A Series of 2,4-Disubstituted Quinolines as a New Class of Allosteric Enhancers of the Adenosine A<sub>3</sub>Receptor Laura H. Heitman, Anikó Göblyös, Annelien J.M. Zweemer, Journal of Medicinal Chemistry	2009	62
Binding Kinetics of ZM241385 Derivatives at the Human Adenosine A<sub>2A</sub> Receptor Dong Guo, Lizi Xia, Jacobus P. D. van Veldhoven, ChemMedChem	2014	49
Development of Covalent Ligands for G Protein-Coupled Receptors: A Case for the Human Adenosine A<sub>3</sub> Receptor Xue Yang, Jacobus P. D. van Veldhoven, Jelle Offringa, Journal of Medicinal Chemistry	2019	44
A new generation of adenosine receptor antagonists: From di- to trisubstituted aminopyrimidines Jacobus P. D. van Veldhoven, Lisa C. W. Chang, Jacobien K. von Frijtag Drabbe Künzel, Bioorganic & Medicinal Chemistry Molecular PharmacologyBiochemistryFunctional SelectivityMedicineReceptor (Biochemistry)	2008	43
Pyrrolone Derivatives as Intracellular Allosteric Modulators for Chemokine Receptors: Selective and Dual-Targeting Inhibitors of CC Chemokine Receptors 1 and 2 Natalia V. Ortiz Zacarı́as, Jacobus P. D. van Veldhoven, Laura Portner, Journal of Medicinal Chemistry	2018	41
Crystal Structure and Subsequent Ligand Design of a Nonriboside Partial Agonist Bound to the Adenosine A<sub>2A</sub> Receptor Tasia Amelia, Jacobus P. D. van Veldhoven, Matteo Falsini, Journal of Medicinal Chemistry	2021	40
Allosteric Modulation of K <sub>v</sub> 11.1 (hERG) Channels Protects Against Drug-Induced Ventricular Arrhythmias Zhiyi Yu, Jia Liu, Jacobus P. D. van Veldhoven, Circulation Arrhythmia and Electrophysiology	2016	34

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