Marco Betti

Design, Synthesis, and Pharmacological Characterization of 2-(2-Furanyl)thiazolo[5,4-<i>d</i>]pyrimidine-5,7-diamine Derivatives: New Highly Potent A_2AAdenosine Receptor Inverse Agonists with Antinociceptive Activity

Flavia Varano, Daniela Catarzi, Fabrizio Vincenzi et al. · Journal of Medicinal Chemistry · 2016 · 57 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

The 1,2,4-Triazolo[4,3-<i>a</i>]pyrazin-3-one as a Versatile Scaffold for the Design of Potent Adenosine Human Receptor Antagonists. Structural Investigations to Target the A_2AReceptor Subtype

Matteo Falsini, Lucia Squarcialupi, Daniela Catarzi et al. · Journal of Medicinal Chemistry · 2017 · 35 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

The aminopyridine-3,5-dicarbonitrile core for the design of new non-nucleoside-like agonists of the human adenosine A2B receptor

Marco Betti, Daniela Catarzi, Flavia Varano et al. · European Journal of Medicinal Chemistry · 2018 · 34 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +10

3-Hydroxy-1<i>H</i>-quinazoline-2,4-dione as a New Scaffold To Develop Potent and Selective Inhibitors of the Tumor-Associated Carbonic Anhydrases IX and XII

Matteo Falsini, Lucia Squarcialupi, Daniela Catarzi et al. · Journal of Medicinal Chemistry · 2017 · 27 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

Exploring the 7-oxo-thiazolo[5,4-d]pyrimidine core for the design of new human adenosine A3 receptor antagonists. Synthesis, molecular modeling studies and pharmacological evaluation

Flavia Varano, Daniela Catarzi, Lucia Squarcialupi et al. · European Journal of Medicinal Chemistry · 2015 · 26 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14