Ester Fernández‐Salas

Discovery of ARD-69 as a Highly Potent Proteolysis Targeting Chimera (PROTAC) Degrader of Androgen Receptor (AR) for the Treatment of Prostate Cancer

Xin Han, Chao Wang, Chong Qin et al. · Journal of Medicinal Chemistry · 2019 · 381 citations · Full text

Medicine, Oncology, Pharmacology +17

Discovery of a Small-Molecule Degrader of Bromodomain and Extra-Terminal (BET) Proteins with Picomolar Cellular Potencies and Capable of Achieving Tumor Regression

Bing Zhou, Jiantao Hu, Fuming Xu et al. · Journal of Medicinal Chemistry · 2017 · 361 citations · Full text

Medicine, Medicinal Chemistry, Oncology +13

Discovery of QCA570 as an Exceptionally Potent and Efficacious Proteolysis Targeting Chimera (PROTAC) Degrader of the Bromodomain and Extra-Terminal (BET) Proteins Capable of Inducing Complete and Durable Tumor Regression

Chong Qin, Yang Hu, Bing Zhou et al. · Journal of Medicinal Chemistry · 2018 · 263 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

Targeted Degradation of BET Proteins in Triple-Negative Breast Cancer

Longchuan Bai, Bing Zhou, Chao‐Yie Yang et al. · Cancer Research · 2017 · 199 citations · Full text

Life Sciences, Oncology, Pharmacology +17

mtCLIC/CLIC4, an Organellular Chloride Channel Protein, Is Increased by DNA Damage and Participates in the Apoptotic Response to p53

Ester Fernández‐Salas, Kwang S. Suh, Vladislav V. Speransky et al. · Molecular and Cellular Biology · 2002 · 188 citations · Full text

Life Sciences, Cell Biology, Pharmacology +17