Aarti Sawant‐Basak

Determination of receptor occupancy in the presence of mass dose: [ ¹¹ C]GSK189254 PET imaging of histamine H ₃ receptor occupancy by PF-03654746

Jean‐Dominique Gallezot, Beata Planeta, Nabeel Nabulsi et al. · Journal of Cerebral Blood Flow & Metabolism · 2016 · 68 citations · Full text

Medicine, Nuclear Medicine, Pharmacology +13

Pharmacological Characterization of 2-Methyl-N-((2′-(pyrrolidin-1-ylsulfonyl)biphenyl-4-yl)methyl)propan-1-amine (PF-04455242), a High-Affinity Antagonist Selective for κ-Opioid Receptors

S. Grimwood, Yang Lü, Anne W. Schmidt et al. · Journal of Pharmacology and Experimental Therapeutics · 2011 · 59 citations

Medicine, Medicinal Chemistry, Pharmacology +14

The 5-Hydroxytryptamine4 Receptor Agonists Prucalopride and PRX-03140 Increase Acetylcholine and Histamine Levels in the Rat Prefrontal Cortex and the Power of Stimulated Hippocampal θ Oscillations

David E. Johnson, Elena M. Drummond, Sarah Grimwood et al. · Journal of Pharmacology and Experimental Therapeutics · 2012 · 57 citations

Medicine, Neuroscience, Pharmacology +16

Quantitative PK–PD Model-Based Translational Pharmacology of a Novel Kappa Opioid Receptor Antagonist Between Rats and Humans

Cheng Chang, Wonkyung Byon, Yifeng Lu et al. · The AAPS Journal · 2011 · 42 citations · Full text

Pharmacy, Pharmacokinetics, Pharmacology +10

Identification of Multiple 5-HT₄Partial Agonist Clinical Candidates for the Treatment of Alzheimer’s Disease

Michael A. Brodney, David E. Johnson, Aarti Sawant‐Basak et al. · Journal of Medicinal Chemistry · 2012 · 42 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17