Mohamed Salah

First Structure–Activity Relationship of 17β-Hydroxysteroid Dehydrogenase Type 14 Nonsteroidal Inhibitors and Crystal Structures in Complex with the Enzyme

Florian Braun, Nicole Bertoletti, Gabriele Möller et al. · Journal of Medicinal Chemistry · 2016 · 30 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Discovery of novel 6-hydroxybenzothiazole urea derivatives as dual Dyrk1A/α-synuclein aggregation inhibitors with neuroprotective effects

Yasmeen T. AlNajjar, Moustafa T. Gabr, Ahmed K. ElHady et al. · European Journal of Medicinal Chemistry · 2021 · 28 citations · Full text

Life Sciences, Medicinal Chemistry, Neuroscience +16

First Dual Inhibitors of Steroid Sulfatase (STS) and 17β-Hydroxysteroid Dehydrogenase Type 1 (17β-HSD1): Designed Multiple Ligands as Novel Potential Therapeutics for Estrogen-Dependent Diseases

Mohamed Salah, Ahmed S. Abdelsamie, Martin Frotscher · Journal of Medicinal Chemistry · 2017 · 25 citations · Full text

Life Sciences, Medicinal Chemistry, Pharmacology +17

Development of novel 2,4-bispyridyl thiophene–based compounds as highly potent and selective Dyrk1A inhibitors. Part I: Benzamide and benzylamide derivatives

Sarah S. Darwish, Mohammad Abdel‐Halim, Mohamed Salah et al. · European Journal of Medicinal Chemistry · 2018 · 24 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

Development of novel amide–derivatized 2,4-bispyridyl thiophenes as highly potent and selective Dyrk1A inhibitors. Part II: Identification of the cyclopropylamide moiety as a key modification

Sarah S. Darwish, Mohammad Abdel‐Halim, Ahmed K. ElHady et al. · European Journal of Medicinal Chemistry · 2018 · 22 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +11