Andrea Ammara

A new framework for novel analogues of pazopanib as potent and selective human carbonic anhydrase inhibitors: Design, repurposing rational, synthesis, crystallographic, in vivo and in vitro biological assessments

Salma M. Hefny, Tarek F. El‐Moselhy, Nabaweya Sharaf El-Din et al. · European Journal of Medicinal Chemistry · 2024 · 35 citations · Full text

Medicinal Chemistry, Vitro Biological Assessments, Biochemistry +11

Discovery of Novel Pyridazine-Tethered Sulfonamides as Carbonic Anhydrase II Inhibitors for the Management of Glaucoma

Haytham O. Tawfik, Mohamed M. Saleh, Andrea Ammara et al. · Journal of Medicinal Chemistry · 2024 · 29 citations · Full text

Discovery of new sulfonamide-tethered 2-aryl-4-anilinoquinazolines as the first-in-class dual carbonic anhydrase and EGFR inhibitors

Wagdy M. Eldehna, Zainab M. Elsayed, Andrea Ammara et al. · International Journal of Biological Macromolecules · 2024 · 14 citations

Combinatorial Chemistry, Medicinal Chemistry, Medicine +10

Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant <i>Neisseria gonorrhoeae</i>

Alessandro Bonardi, Alessio Nocentini, Simone Giovannuzzi et al. · Journal of Medicinal Chemistry · 2024 · 12 citations · Full text

Development of novel anilinoquinazoline-based carboxylic acids as non-classical carbonic anhydrase IX and XII inhibitors

Zainab M. Elsayed, Hadia Almahli, Alessio Nocentini et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 2023 · 11 citations · Full text