Goss S. Kauffman

An Efficient Chiral Moderator Prepared from Inexpensive (+)-3-Carene:  Synthesis of the HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitor DPC 963

Goss S. Kauffman, Gregory D. Harris, Roberta L. Dorow et al. · Organic Letters · 2000 · 193 citations

Bioorganic Chemistry, Molecular Biology, Chiral Moderator +19

Rearrangement of N_α-Protected <scp>l</scp>-Asparagines with Iodosobenzene Diacetate. A Practical Route to β-Amino-<scp>l</scp>-alanine Derivatives

Linhua Zhang, Goss S. Kauffman, Jaan A. Pesti et al. · The Journal of Organic Chemistry · 1997 · 98 citations

Organic Chemistry, Peptide Science, Protected Asparagines +17

Synthesis and structure based optimization of novel Akt inhibitors

Blaise Lippa, Gonghua Pan, Matthew S. Corbett et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 74 citations · Full text

Medicinal Chemistry, Medicine, Rational Drug Design +5

Synthesis of Thrombin Inhibitor DuP 714

John Wityak, Richard A. Earl, Matthew M. Abelman et al. · The Journal of Organic Chemistry · 1995 · 74 citations

Altmetric Attention Score, Pharmacotherapy, Chemical Biology +18

Discovery and Optimization of Quinolinone Derivatives as Potent, Selective, and Orally Bioavailable Mutant Isocitrate Dehydrogenase 1 (mIDH1) Inhibitors

Jian Lin, Wei Lu, Justin A. Caravella et al. · Journal of Medicinal Chemistry · 2019 · 46 citations · Full text