Jeffrey K. Kerns

Monoacidic Inhibitors of the Kelch-like ECH-Associated Protein 1: Nuclear Factor Erythroid 2-Related Factor 2 (KEAP1:NRF2) Protein–Protein Interaction with High Cell Potency Identified by Fragment-Based Discovery

Thomas G. Davies, William E. Wixted, Joseph E. Coyle et al. · Journal of Medicinal Chemistry · 2016 · 306 citations · Full text

Life Sciences, Medicinal Chemistry, Pharmacology +17

Structure of the BTB Domain of Keap1 and Its Interaction with the Triterpenoid Antagonist CDDO

Anne Cleasby, Jeff Yon, Philip J. Day et al. · PLoS ONE · 2014 · 254 citations · Full text

Life Sciences, Biochemistry, Molecular Biology +17

Keap Calm, and Carry on Covalently

A. James Wilson, Jeffrey K. Kerns, James F. Callahan et al. · Journal of Medicinal Chemistry · 2013 · 170 citations

Life Sciences, Biochemistry, Pharmacology +17

Growth Inhibition of Hepatoma Cells Induced by Vitamin K and Its Analogs

Yuji Nishikawa, Brian I. Carr, Meifang Wang et al. · Journal of Biological Chemistry · 1995 · 141 citations · Full text

Life Sciences, Biochemistry, Cell Biology +9

The Spongistatins: Architecturally Complex Natural Products-Part Two: Synthesis of the C(29-51) Subunit, Fragment Assembly, and Final Elaboration to (+)-Spongistatin 2

Amos B. Smith, Qiyan Lin, Victoria A. Doughty et al. · Angewandte Chemie International Edition · 2001 · 108 citations

Natural Sciences, Chemistry, Molecular Biology +12