Concepedia

Optimization of a novel series of N-phenylindoline-5-sulfonamide-based acyl CoA:monoacylglycerol acyltransferase-2 inhibitors: Mitigation of CYP3A4 time-dependent inhibition and phototoxic liabilities

Kenjiro Sato, Hiroki Takahagi, Osamu Kubo, Kousuke Hidaka, Takeshi Yoshikawa, Masahiro Kamaura, Masanori Nakakariya, Nobuyuki Amano, Ryutaro Adachi, Toshiyuki Maki,

Bioorganic & Medicinal Chemistry · 2015 · 11 citations · 27 references

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27

A short history of<i>SHELX</i>

George M. Sheldrick · Acta Crystallographica Section A Foundations of Crystallography · 2007 · 87.4K citations · Full text

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Development and use of quantum mechanical molecular models. 76. AM1: a new general purpose quantum mechanical molecular model

Michael J. S. Dewar, Eve G. Zoebisch, Eamonn F. Healy et al. · Journal of the American Chemical Society · 1985 · 13.1K citations

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Nonfasting Triglycerides and Risk of Myocardial Infarction, Ischemic Heart Disease, and Death in Men and Women

Børge G. Nordestgaard, Marianne Benn, Peter Schnohr et al. · JAMA · 2007 · 2.1K citations

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Cloning of DGAT2, a Second Mammalian Diacylglycerol Acyltransferase, and Related Family Members

Sylvaine Cases, Scot J. Stone, Ping Zhou et al. · Journal of Biological Chemistry · 2001 · 801 citations · Full text

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A New Class of Easily Activated Palladium Precatalysts for Facile C−N Cross-Coupling Reactions and the Low Temperature Oxidative Addition of Aryl Chlorides

Mark R. Biscoe, Brett P. Fors, Stephen L. Buchwald · Journal of the American Chemical Society · 2008 · 415 citations · Full text

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